Melanotan II · DOSSIER

Melanotan II

MT-2 · MT-II · Peptide · 7 AS
LEGAL DE · NOT APPROVEDEVIDENCE · PRECLINICAL2 STUDIESWADA · S2
SUMMARY

Prompts the skin cells to produce more pigment (melanin) — the skin darkens, even with little sun.

FIG.01 — SIGNAL CHAIN
Ac-Nle-cyclo[Asp-His-D-Phe-Arg-Trp-Lys]-NH₂ · ~1024.2 Da
EVIDENCE LEVELSPROVEN IN HUMANSANIMAL MODELS ONLYMECHANISM ONLYUNPROVEN IN HUMANS
01

What it does in the body

Findings, each with its evidence level — animal data kept visibly apart from what's unproven in humans.

Tans the skin

Prompts the skin cells to produce more pigment (melanin) — the skin darkens, even with little sun.

PROVEN IN HUMANS
May boost libido & erection

Acts on sexual desire in the brain; early studies showed such effects (later developed further as PT-141).

PROVEN IN HUMANS
Not approved — with serious risks

Not approved as a drug anywhere; dermatologists report melanoma cases and sometimes strong blood-pressure spikes.

UNPROVEN IN HUMANS
02

Mechanism of action

What Melanotan II does in the body — step by step.

01

Melanotan II is a synthetic cyclic heptapeptide and a non-selective agonist at melanocortin receptors (MC1R, MC3R, MC4R, MC5R).

02

Activation of MC1R in melanocytes stimulates melanin synthesis, leading to increased skin pigmentation.

03

MC4R activation in the hypothalamus is associated with effects on sexual desire and erectile mechanisms.

03

Research status

How far along is the evidence?

PRECLINICALEARLY CLINICAL STUDIESCLINICALLY ESTABLISHED
Melanotan II was originally investigated at the University of Arizona in the context of melanoma prevention and erectile dysfunction.
Melanotan II was originally investigated at the University of Arizona in the context of melanoma prevention and erectile dysfunction.
Early clinical Phase I/II studies documented pigmentation effects and pro-erectile actions.
Clinical development was not continued; instead, PT-141 was developed as a more selective and better tolerated successor.
Since the early 2000s, MT-2 has circulated as an unapproved substance on grey and black markets.
Systematic current safety data on commercial preparations are lacking; reports of increased melanoma under MT-2 use are described in the dermatological literature.
04

Known risks

Without human data, safety statements are limited. What is known:

01
Melanoma risk: repeatedly described cases of activation of pre-existing naevi and melanoma development under MT-2 use in the dermatological literature
02
Hypertension: frequent and sometimes pronounced increases in blood pressure
03
Nausea, vomiting, flushing (frequent)
04
Unwanted spontaneous erections (reported from clinical studies)
05
Irreversible hyperpigmentation possible
06
Product quality cannot be verified from illegal sources — contaminants and incorrect dosages documented
07
BfArM and MHRA have issued explicit safety warnings
05

Cited studies

Chronological — links lead to the source.

1996
Activation of melanocortin receptors in vitro and in vivo by MT-II
PubMed 8930207 →
1998
Melanotan II, a melanocortin receptor agonist, increases penile erection in men
PubMed 9544831 →
06

Frequently asked questions

What is Melanotan II?+

Melanotan II is a synthetic cyclic heptapeptide and a non-selective agonist at melanocortin receptors (MC1R, MC3R, MC4R, MC5R).

What type of peptide is Melanotan II?+

Melanotan II belongs to the Melanocortin class.

What is Melanotan II used for?+

In research, Melanotan II has primarily been investigated in the context of: Libido, Skin & hair. These are research findings (evidence: preclinical), not proven benefits in humans and not a usage recommendation.

Is Melanotan II legal in Germany?+

Melanotan II is not approved as a medicine in Germany. Obtaining it outside clinical studies is legally problematic.

Is Melanotan II FDA-approved / legal in the US?+

No. Melanotan II is not FDA-approved as a drug in the US; it is mostly sold as a research chemical and not for human consumption.

Is Melanotan II legal in Canada?+

No. Melanotan II is not authorized by Health Canada and not intended for human consumption.

Where can I buy Melanotan II?+

Peptica sells nothing and names no sources. Melanotan II is "not approved" in Germany; obtaining unapproved substances outside clinical studies is illegal and carries quality and safety risks.

What is the dosage of Melanotan II?+

Peptica publishes no dosing. There are no approved dosing guidelines for Melanotan II; figures circulating online stem from animal studies or anecdote, not from validated human protocols. This is not medical advice.

Is Melanotan II banned in sport (WADA)?+

Yes. Melanotan II is on the WADA Prohibited List and is therefore banned in competitive sport.

What are the known risks of Melanotan II?+

Documented risks include: Melanoma risk: repeatedly described cases of activation of pre-existing naevi and melanoma development under MT-2 use in the dermatological literature; Hypertension: frequent and sometimes pronounced increases in blood pressure. This is not a complete safety assessment and not medical advice — see the risks section for the full list.

How well researched is Melanotan II?+

The evidence is classified as “preclinical”. 2 studies are cited on this page.

What is the molecular weight of Melanotan II?+

Melanotan II has a molar mass of about 1024.2 Da.

Which peptides are related to Melanotan II?+

Closely related entries: PT-141. A direct side-by-side comparison is available via the compare function.

07

Dossier

Legal · Structure · Sources.

LEGAL STATUS BY REGION
Germanynot approved

Melanotan II is on the WADA Prohibited List (S4: hormones and metabolic modulators). It is not approved as a medicine in the EU, Germany, Austria or Switzerland. Several European authorities (MHRA in the UK, BfArM in Germany) have issued explicit warnings about MT-2, highlighting considerable safety risks. Possession and import are problematic in Germany under the AMG; for athletes, the ADBG additionally applies. The EU Commission has added MT-2 to warning lists for dangerous substances.

Legal status varies by country and can change. This is not legal advice.

STRUCTURE & MOLECULE
H₂NAc-Nle-cyclo[Asp-His-D-Phe-Arg-Trp-Lys]-NHCOOH
7
AMINO ACIDS
~1024.2
MOL. WEIGHT (Da)
Limited data; the plasma half-life is reported to be around one hour (sources range from ~30 minutes to a few hours)
HALF-LIFE
SOURCES & EXTERNAL DATABASES

Methodology: Peptica compiles publicly available studies and regulatory information and assigns each statement an evidence level. Not medical advice. No warranty.

RELATED PEPTIDES & FURTHER READING
08

Community notes

Note: These posts are user opinions and not medical advice. Posts containing dosages, therapeutic claims or purchase recommendations are removed. All entries are manually reviewed before publication.
This page is intended solely for factual, scientifically oriented information. No medical advice · no dosage or usage recommendations · no claims of efficacy · no substitute for medical consultation. Peptica sells no substances. Partner links are marked as advertising; Peptica may earn a commission. © 2026 Peptica · Issue 01